| 货号:30602-1 mg | 规格:1 mg | 目录价:¥925 |
| 货号:30602-10 mg | 规格:10 mg | 目录价:¥3122 |
| 货号:30602-25 mg | 规格:25 mg | 目录价:¥6606 |
| 货号:30602-5 mg | 规格:5 mg | 目录价:¥1769 |
产品详情
* 以下信息仅供参考,详情请以原厂网站为准
产品名称:
ADTL-EI1712
产品描述:
A dual ERK1 and ERK5 inhibitor (IC50s = 40.43 and 64.5 nM, respectively); reduces ERK1 and ERK5 activity by 93.5% and 89.4%, respectively, but also inhibits ERK2 activity by 92.7%, in a panel of 100 kinases at 1 µM; inhibits proliferation of HL-60 and MKN74 cancer cells (IC50s = 1.26 and 2.55 µM, respectively); reduces tumor growth and intratumor phosphorylation of ERK1/2 and ERK5 in an MKN74 mouse xenograft model at 50 mg/kg per day
保存温度:
-20
运输温度:
-20
预期分子量:
505.44148
产品形式:
A crystalline solid
纯度:
≥98%
CAS号:
2414916-45-1
分子式:
C22H18Cl2N4O2S2
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