AH 6809-激动剂-深圳欣博盛生物科技有限公司

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AH 6809

品牌：Cayman

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说明书

折扣/货期

货号：14050-1 mg	规格：1 mg	目录价：￥281
货号：14050-10 mg	规格：10 mg	目录价：￥2037
货号：14050-5 mg	规格：5 mg	目录价：￥1152
货号：14050-50 mg	规格：50 mg	目录价：￥8777

产品详情

* 以下信息仅供参考，详情请以原厂网站为准

产品名称:

AH 6809

产品描述:

AH 6809 is an EP and DP receptor antagonist with nearly equal affinity for the cloned human EP1, EP2, EP3-III, and DP1 receptors.{8322} AH 6809 blocks the PGE2-induced accumulation of cAMP in COS cells transfected with the human EP2 receptor.{3391} It also blocks the accumulation of Ca2+ in Xenopus oocytes expressing the human EP1 receptor.{3176} In the human and guinea pig, the activity profile of AH 6809 is similar to that of SC-19220, but it is somewhat more potent.{3409} In the mouse, AH 6809 has the highest affinity for the EP2 receptor, but also acts as a weak ligand at the murine EP1 and DP1 receptors.{6640} In whole human platelets, AH 6809 is an effective antagonist of the antiaggregatory actions of PGD2, but not PGI2, with an EC50 of about 5 x 10−5 M.{3319}

保存温度:

-20

运输温度:

-20

预期分子量:

298.3

产品形式:

A crystalline solid

纯度:

≥97%

CAS号:

33458-93-4