深圳欣博盛生物科技有限公司 a1

Amantadine (hydrochloride)
货号:21364-10 g 规格:10 g 目录价:¥482
货号:21364-100 g 规格:100 g 目录价:¥2935
货号:21364-25 g 规格:25 g 目录价:¥884
货号:21364-50 g 规格:50 g 目录价:¥1608
产品详情
* 以下信息仅供参考,详情请以原厂网站为准
产品名称:
Amantadine (hydrochloride)
别名:
Adamantylamine|Aminoadamantane|NSC 83653
产品描述:
An NMDAR antagonist (IC50s = 0.93, 0.82, and 0.47 μM at -70 mV for NR1-1a/NR2A, NR1-1a/NR2B, and NR1-1a/NR2D subunit-containing recombinant receptors, respectively, expressed in HEK293 cells); blocks the influenza A M2 proton channel (IC50 = 16 μM for the recombinant channel expressed in Xenopus oocytes) and inhibits cytotoxicity induced by the influenza A strains H1N1 and H3N2 in MDCK cells (EC50s = 34 and 0.84 μM, respectively); improves the survival of mice infected with influenza A when administered 24 hours following viral challenge at a dose of 100 mg/kg per day; decreases L-DOPA-induced dyskinesia in a 6-OHDA hemi-parkinsonian mouse model at 40 mg/kg
保存温度:
-20
运输温度:
-20
预期分子量:
151.24
产品形式:
A crystalline solid
纯度:
≥95%
CAS号:
665-66-7
分子式:
C10H17N • HCl
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