| 货号:21299-1 mg | 规格:1 mg | 目录价:¥844 |
| 货号:21299-10 mg | 规格:10 mg | 目录价:¥3739 |
| 货号:21299-5 mg | 规格:5 mg | 目录价:¥2090 |
产品详情
* 以下信息仅供参考,详情请以原厂网站为准
产品名称:
ARV-771
产品描述:
A PROTAC that drives BET family protein degradation; induces degradation of BRD2, BRD3, and BRD4 in 22Rv1 CRPC cells (DC50s = <5 nM for all); inhibits proliferation of and increases PARP cleavage in 22Rv1 cells in a concentration-dependent manner; reduces full-length androgen receptor protein levels and prevents R1881-induced increases in ERG in VCaP cells; induces tumor regression in a 22Rv1 mouse xenograft model at 30 mg/kg per day, s.c.
保存温度:
-20
运输温度:
-20
预期分子量:
986.6
产品形式:
A crystalline solid
纯度:
≥95%
CAS号:
1949837-12-0
分子式:
C49H60ClN9O7S2
促销活动
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