| 货号:44842-10 mg | 规格:10 mg | 目录价:¥1273 |
| 货号:44842-25 mg | 规格:25 mg | 目录价:¥2653 |
| 货号:44842-5 mg | 规格:5 mg | 目录价:¥1059 |
| 货号:44842-50 mg | 规格:50 mg | 目录价:¥4770 |
产品详情
* 以下信息仅供参考,详情请以原厂网站为准
产品名称:
ATX968
别名:
DHX9 Inhibitor 2|DHX9-IN-2
产品描述:
A DDX9 inhibitor (IC50 = 8 nM for helicase activity); selective for DDX9 over DDX36, BRM, and WRN (IC50s = >10, >10, and >100 µM, respectively), as well as a panel of 96 kinases at 10 µM but does inhibit DYRK1B; selectively induces unresolved nuclear R-loop accumulation in MSI-H/dMMR LS411N colorectal carcinoma cells over MSS/pMMR NCI H747 colorectal carcinoma cells at 1 µM; induces tumor regression in an LS411N mouse xenograft model at 300 mg/kg
保存温度:
-20
运输温度:
-20
预期分子量:
421.914
产品形式:
A solid
纯度:
≥98%
CAS号:
2973395-71-8
分子式:
C18H16ClN3O3S2
促销活动
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官网链接
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