深圳欣博盛生物科技有限公司 a1

AVN-101 (hydrochloride)
货号:38791-1 mg 规格:1 mg 目录价:¥442
货号:38791-10 mg 规格:10 mg 目录价:¥1755
货号:38791-25 mg 规格:25 mg 目录价:¥3296
货号:38791-5 mg 规格:5 mg 目录价:¥992
产品详情
* 以下信息仅供参考,详情请以原厂网站为准
产品名称:
AVN-101 (hydrochloride)
产品描述:
A multimodal receptor antagonist; an antagonist of 5-HT7, 5-HT2C, 5-HT2A, and 5-HT6 receptors (Kis = 0.153, 1.17, 1.56, and 2.04 nM, respectively); selective for these receptors over 5-HT2B, 5-HT5A, 5-HT1A, and 5-HT1B receptors (Kis = 10.6, 20.8, 61, and 720 nM, respectively); an antagonist of α2A-, α2B-, α2C-, α1B-, α1A-, and α1D-adrenergic receptors (Kis = 0.41, 1.77, 3.55, 9.4, 18.9, and 30.2 nM, respectively), as well as histamine H1 and H2 receptors (Kis = 0.58 and 89 nM, respectively); increases the time spent in the open arms of the elevated plus maze in mice at 0.2, 1, and 5 mg/kg; reduces immobility in the forced swim test and prevents scopolamine-induced amnesia in a passive avoidance test in mice at 0.05 mg/kg
保存温度:
-20
运输温度:
-20
预期分子量:
304.42874
产品形式:
A crystalline solid
纯度:
≥98%
CAS号:
1061354-48-0
分子式:
C21H24N2 • HCl
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