| 货号:22932-1 mg | 规格:1 mg | 目录价:¥429 |
| 货号:22932-10 mg | 规格:10 mg | 目录价:¥2117 |
| 货号:22932-25 mg | 规格:25 mg | 目录价:¥3685 |
| 货号:22932-5 mg | 规格:5 mg | 目录价:¥1273 |
产品详情
* 以下信息仅供参考,详情请以原厂网站为准
产品名称:
BIBS39
产品描述:
A nonpeptide AT1 receptor antagonist (Ki = 29 nM in rat lung membranes); selective for AT1 over AT2 receptors (Ki = 480 nM in isolated rat adrenal medulla), as well as α1-, α2-, β1-, and β2-adrenergic, adenosine A1 and A2, muscarinic M1, M2, and M3, and atrial natriuretic peptide receptors (Kis = >100 µM for all); decreases diastolic blood pressure in pithed normotensive rats without affecting heart rate at 0.3-10 mg/kg; decreases diastolic blood pressure in renal hypertensive rats with an increase in heart rate at 1-30 mg/kg
保存温度:
-20
运输温度:
-20
预期分子量:
524.7
产品形式:
A crystalline solid
纯度:
≥98%
CAS号:
133085-33-3
分子式:
C32H36N4O3
促销活动
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