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折扣/货期| 货号：31446-1 mg | 规格：1 mg | 目录价：￥482.4 |
| 货号：31446-10 mg | 规格：10 mg | 目录价：￥3591.2 |
| 货号：31446-25 mg | 规格：25 mg | 目录价：￥7865.8 |
| 货号：31446-5 mg | 规格：5 mg | 目录价：￥2050.2 |
产品详情
* 以下信息仅供参考，详情请以原厂网站为准
产品名称:
Cariprazine
别名:
RGH-188
产品描述:
An atypical antipsychotic; binds to dopamine D2L, D2S, and D3, 5-HT1A, 5-HT2A, 5-HT2B, histamine H1, and σ1 receptors (Kis = 0.085-23.44 nM); an antagonist of dopamine D2 and D3 receptors (Kbs = 0.759 and 0.316 nM, respectively); a partial agonist at dopamine D2 and D3 receptors; stimulates inositol phosphate production in murine A9 cells expressing human D2L receptors (EC50 = 3.16 nM); inhibits forskolin-induced cAMP accumulation in CHO cells expressing human D3 receptors (EC50 = 2.63 nM); inhibits amphetamine-induced hyperactivity and the conditioned avoidance response in rats (ED50s = 0.12 and 0.84 mg/kg, respectively); inhibits scopolamine-induced learning deficits in a water labyrinth learning test in rats from 0.02-0.08 mg/kg
保存温度:
-20
运输温度:
-20
预期分子量:
427.41054
产品形式:
A crystalline solid
有效期:
1460
纯度:
≥95%
CAS号:
839712-12-8
分子式:
C21H32Cl2N4O
促销活动
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