深圳欣博盛生物科技有限公司 a1

Carvedilol
货号:15418-100 mg 规格:100 mg 目录价:¥询价
货号:15418-250 mg 规格:250 mg 目录价:¥询价
货号:15418-50 mg 规格:50 mg 目录价:¥询价
产品详情
* 以下信息仅供参考,详情请以原厂网站为准
产品名称:
Carvedilol
别名:
BM 14190
产品描述:
A β-adrenergic receptor antagonist (Kds = 1.78, 0.4, and 5.01 nM for β1-, β2-, and β3-ARs, respectively); selectively binds to α1- over α2-ARs (Kis = 0.81 and 3,400 nM, respectively); reverses increases in heart rate induced by isoproterenol in isolated guinea pig atria (Kb = 0.8 nM); prevents epinephrine-induced premature ventricular beats in a rat model of arrhythmia (ED50 = 0.25 mg/kg); inhibits the contractile response to norepinephrine in isolated rabbit aorta (Kb = 11 nM); decreases systolic blood pressure and heart rate in rat models of hypertension from 3-30 mg/kg; inhibits SARS-CoV-2 Mpro (IC50 = 204.6 µg/ml) and reduces viral infectivity in SARS-CoV-2-infected Vero E6 cells (IC50 = 0.350 µg/ml)
保存温度:
-20
运输温度:
-20
预期分子量:
406.5
产品形式:
A crystalline solid
纯度:
≥98%
CAS号:
72956-09-3
分子式:
C24H26N2O4
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