货号:43519-1 mg | 规格:1 mg | 目录价:¥812 |
货号:43519-10 mg | 规格:10 mg | 目录价:¥2842 |
货号:43519-5 mg | 规格:5 mg | 目录价:¥1624 |
产品详情
* 以下信息仅供参考,详情请以原厂网站为准
产品名称:
CM699 (hydrochloride)
产品描述:
A dual σ receptor antagonist (Kis = 0.0141 and 0.00231 µM for the σ1 and σ2 receptors, respectively) and DAT inhibitor (Ki = 0.311 µM); selective for the σ1 and σ2 receptors and DAT over SERT (Ki = 2.83 µM) but also binds to NET (Ki = 0.232 µM); inhibits dopamine uptake in rat striatal synaptosomes (IC50 = 6.01 µM) and induces σ1 receptor multimerization, indicating antagonist activity, in HEK293 cells expressing the human receptor at 20 µM; decreases self-administration of cocaine in rats
保存温度:
-20
运输温度:
-20
预期分子量:
427.973
产品形式:
A neat solid
有效期:
1460
纯度:
≥98%
分子式:
C24H29N3O2 • HCl
促销活动
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