| 货号:19915-1 mg | 规格:1 mg | 目录价:¥询价 |
| 货号:19915-10 mg | 规格:10 mg | 目录价:¥询价 |
| 货号:19915-25 mg | 规格:25 mg | 目录价:¥询价 |
| 货号:19915-5 mg | 规格:5 mg | 目录价:¥询价 |
产品详情
* 以下信息仅供参考,详情请以原厂网站为准
产品名称:
Daprodustat
别名:
GSK1278863
产品描述:
A HIF-PH1, -2, and -3 inhibitor (IC50s = 3.5, 22.2, 5.5 nM, respectively); selective for HIF-PH1, -2, and -3 over FIH and CP4H (IC50s = 9,800 and >200,000 nM, respectively); induces accumulation of HIF-1α and HIF-2α in Hep3B cells at 25 and 50 µM; increases plasma levels of EPO in mice at 60 mg/kg; increases the number of reticulocytes and levels of hemoglobin in mice at 3, 10, and 30 mg/kg
保存温度:
-20
运输温度:
-20
预期分子量:
393.4
产品形式:
A crystalline solid
有效期:
1460
纯度:
≥98%
CAS号:
960539-70-2
分子式:
C19H27N3O6
促销活动
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