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折扣/货期| 货号：27636-1 mg | 规格：1 mg | 目录价：￥871 |
| 货号：27636-10 mg | 规格：10 mg | 目录价：￥3484 |
| 货号：27636-25 mg | 规格：25 mg | 目录价：￥6539 |
| 货号：27636-5 mg | 规格：5 mg | 目录价：￥2184 |
产品详情
* 以下信息仅供参考，详情请以原厂网站为准
产品名称:
Derazantinib
别名:
ARQ 087
产品描述:
A multi-kinase inhibitor; a pan inhibitor of FGFR (IC50s = 4.5, 1.8, 4.5, and 34 nM for FGFR1, -2, -3, and -4, respectively); inhibits 18 tyrosine kinases and the calcium/calmodulin-dependent protein kinase QIK in a panel of 297 kinases (IC50s = 3-31 and 9.7 nM, respectively); decreases phosphorylation of FGFR in COS-1 cells expressing FGFR1, -2, -3, or -4 (IC50s = 10 µM, respectively) and inhibits the growth of 15 cancer cell lines with mutant, amplified, or translocated FGFR (GI50s = 0.1-1.7 µM); reduces tumor growth and decreases tumor protein levels of phosphorylated FGFR, FRS2, and ERK in a SNU-16 mouse xenograft model at 50 and 75 mg/kg
保存温度:
-20
运输温度:
-20
预期分子量:
468.565323
产品形式:
A crystalline solid
纯度:
≥95%
CAS号:
1234356-69-4
分子式:
C29H29FN4O
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