深圳欣博盛生物科技有限公司 a1

Efaroxan (hydrochloride)
货号:29008-10 mg 规格:10 mg 目录价:¥549
货号:29008-25 mg 规格:25 mg 目录价:¥1072
货号:29008-50 mg 规格:50 mg 目录价:¥1447
产品详情
* 以下信息仅供参考,详情请以原厂网站为准
产品名称:
Efaroxan (hydrochloride)
别名:
(±)-Efaroxan|RX-821037
产品描述:
An α2-AR (EC50s = 1 receptor antagonist; binds to α2A-, α2B-, and α2C-ARs (Kis = 13, 38, and 1,820 nM, respectively) and selectively to I1 over I2 receptors (Kis = 52 and >10,000 nM, respectively); binds to putative I3 receptors on human pancreatic islets of Langerhans and stimulates insulin secretion at 100 μM; binds to rat RIN-5AH insulinoma cell membranes (IC50g = 32 nM) and stimulates insulin secretion at 100 μM; lowers basal blood glucose levels in mice at 5 mg/kg; increases L-DOPA synthesis in rat cortex and hippocampus by 77 and 57%, respectively at 10 mg/kg
保存温度:
-20
运输温度:
-20
预期分子量:
216.27902
产品形式:
A solid
纯度:
≥98%
CAS号:
89197-00-2
分子式:
C13H16N2O • HCl
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