深圳欣博盛生物科技有限公司 a1

Elagolix (sodium salt)
货号:26534-10 mg 规格:10 mg 目录价:¥2117
货号:26534-25 mg 规格:25 mg 目录价:¥4677
货号:26534-5 mg 规格:5 mg 目录价:¥1206
产品详情
* 以下信息仅供参考,详情请以原厂网站为准
产品名称:
Elagolix (sodium salt)
产品描述:
An antagonist of GnRHR (Ki = 0.9 nM in a radioligand binding assay); selective for GnRHR over CYP3A4 (IC50 = 56 μM) as well as a panel of 100 receptors, ion channels, enzymes, and transporters (IC50s = >10 μM); inhibits GnRH-induced inositol phosphate production in RBL-1 cells expressing human GnRHR (IC50 = 1.5 nM); suppresses production of luteinizing hormone in castrated male cynomolgus macaques at 30 mg/kg
保存温度:
-20
运输温度:
-20
预期分子量:
630.581896
产品形式:
A crystalline solid
纯度:
≥98%
CAS号:
832720-36-2
分子式:
C32H29F5N3O5 • Na
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