深圳欣博盛生物科技有限公司 a1

Endomorphin 2 (trifluoroacetate salt)
货号:23281-1 mg 规格:1 mg 目录价:¥482
货号:23281-5 mg 规格:5 mg 目录价:¥1715
产品详情
* 以下信息仅供参考,详情请以原厂网站为准
产品名称:
Endomorphin 2 (trifluoroacetate salt)
别名:
Tyr-Pro-Phe-Phe-NH2
产品描述:
An endogenous neuropeptide and μ-opioid receptor agonist (Ki = 0.69 nM); selective for μ- over δ- and κ-opioid receptors (Kis = 9,233 and 5,240 nM, respectively); binds to mouse brain membranes and rat recombinant μ-opioid receptors expressed in CHO cells (Kis = 1.37 and 0.58 nM, respectively); inhibits forskolin-induced cAMP accumulation in CHO cells expressing rat recombinant μ-opioid receptors and in SH-SY5Y human neuroblastoma cells (IC50s = 7.08 and 7.76 nM, respectively); increases analgesia in a radiant heat tail-flick assay in mice following intracerebroventricular or intrathecal administration (ED50s = 1.99 and 3.81 μg, respectively); induces conditioned place aversion in mice at 10 μg, i.c.v.; decreases gastrointestinal transit time in mice at 3 μg, i.c.v.
保存温度:
-20
运输温度:
-20
预期分子量:
571.66688
产品形式:
A lyophilized powder
纯度:
≥95%
分子式:
C32H37N5O5 • XCF3COOH
在线留言
咨询类型
联系人
*
联系方式
*
单位名称
*
咨询内容
*
复制QQ号成功,请打开QQ后添加好友进行咨询