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折扣/货期| 货号：23670-10 mg | 规格：10 mg | 目录价：￥2251.2 |
| 货号：23670-100 mg | 规格：100 mg | 目录价：￥11644.6 |
| 货号：23670-5 mg | 规格：5 mg | 目录价：￥1206 |
| 货号：23670-50 mg | 规格：50 mg | 目录价：￥7008.2 |
产品详情
* 以下信息仅供参考，详情请以原厂网站为准
产品名称:
Evacetrapib
产品描述:
A benzazepine-based inhibitor of CETP (IC50s = 5.5 and 26 nM for human recombinant and plasma-derived proteins, respectively); selective for CETP over a panel of cell surface and nuclear receptors at 1 µM; reduces expression of PCSK9 and LDLR in HepG2 cells in a dose-dependent manner; reduces protein levels of LDLR, SREBF2-M, and PCSK9 in HepG2 lysates, nuclear extracts, and culture medium, respectively, in a dose-dependent manner; inhibits CETP activity by 98.5, 98.6, and 18.4% at four, eight, and 24 h, respectively, in CETP/ApoA1 transgenic mice at 30 mg/kg; increases HDL cholesterol levels in serum from CETP/ApoA1 transgenic mice in a dose-dependent manner, including by 129.7% eight hours after a 30 mg/kg dose
保存温度:
-20
运输温度:
-20
预期分子量:
638.7
产品形式:
A crystalline solid
有效期:
1460
纯度:
≥98%
CAS号:
1186486-62-3
分子式:
C31H36F6N6O2
促销活动
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