| 货号:36555-1 mg | 规格:1 mg | 目录价:¥482 |
| 货号:36555-10 mg | 规格:10 mg | 目录价:¥2332 |
| 货号:36555-25 mg | 规格:25 mg | 目录价:¥5226 |
| 货号:36555-5 mg | 规格:5 mg | 目录价:¥1286 |
产品详情
* 以下信息仅供参考,详情请以原厂网站为准
产品名称:
FIT-039
产品描述:
A Cdk9 inhibitor (IC50 = 5.8 µM for Cdk9/cyclin T1); selective for Cdk9/cyclin T1 over Cdk4/cyclin D3 at 30 µM and Cdk2/cyclin A2, Cdk2/cyclin E1, Cdk5/p25, Cdk6/cyclin D3, and Cdk7/cyclin/MAT1 at 10 µM; inhibits GSK3α, GSK3β, PKN1, haspin, p70S6K, DYRK1B, DYRK3, and IRR at 10 µM; inhibits DNA replication of HSV-1 in HeLa cells (IC50 = 0.69 µM); reduces skin lesions and improves survival in HSV-1-infected mice when applied topically at 1.25-10% w/w; reduces tumor growth in an HPV type 16-positive Ca Ski cervical cancer mouse xenograft model at 300 mg/kg
保存温度:
-20
运输温度:
-20
预期分子量:
315.409443
产品形式:
A solid
纯度:
≥98%
CAS号:
1113044-49-7
分子式:
C17H18FN3S
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