| 货号:36601-1 mg | 规格:1 mg | 目录价:¥589.6 |
| 货号:36601-10 mg | 规格:10 mg | 目录价:¥4073.6 |
| 货号:36601-25 mg | 规格:25 mg | 目录价:¥5802.2 |
| 货号:36601-5 mg | 规格:5 mg | 目录价:¥2184.2 |
产品详情
* 以下信息仅供参考,详情请以原厂网站为准
产品名称:
GDC-046
产品描述:
A TYK2 inhibitor (Ki = 4.8 nM); selective for TYK2 over JAK1, -2, and -3 (Kis = 83.8, 27.6, and 253 nM, respectively); selectively inhibits TYK2-mediated IL-12-induced phosphorylation of STAT4 over JAK1-mediated IL-6-induced phosphorylation of STAT3 and JAK2-mediated erythropoietin-induced phosphorylation of STAT5 in cell-based assays (EC50s = 380, 2,000, and 1,700 nM, respectively)
保存温度:
-20
运输温度:
-20
预期分子量:
350.19884
产品形式:
A solid
有效期:
1460
纯度:
≥98%
CAS号:
1258292-64-6
分子式:
C16H13Cl2N3O2
促销活动
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