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折扣/货期| 货号：36705-10 mg | 规格：10 mg | 目录价：￥2907.8 |
| 货号：36705-25 mg | 规格：25 mg | 目录价：￥5641.4 |
| 货号：36705-5 mg | 规格：5 mg | 目录价：￥1621.4 |
产品详情
* 以下信息仅供参考，详情请以原厂网站为准
产品名称:
GSK189254
别名:
GSK189254A
产品描述:
A histamine H3 receptor antagonist (Kis = 0.13, 0.68, and 1.74 nM for the recombinant human, rat, and mouse receptors, respectively); selective for the histamine H3 receptor over a panel of 50 receptors and ion channels at 1 µM; prevents imetit-induced decreases in forskolin-stimulated cAMP accumulation in HEK293-Gαo cells expressing the human histamine H3 receptor (pA2 = 9.06); inhibits intake R-(–)-α-methylhistamine-induced increases in water intake and reverses scopolamine-induced memory deficits in the passive avoidance test in rats; increases hindlimb grip force in a rat model of monoiodoacetate-induced osteoarthritic pain and increases the paw withdrawal threshold in a rat model of spinal nerve ligation-induced neuropathic pain (ED50s = 0.77 and 1.5 mg/kg, i.p., respectively)
保存温度:
-20
运输温度:
-20
预期分子量:
351.44222
产品形式:
A solid
有效期:
1460
纯度:
≥98%
CAS号:
720690-73-3
分子式:
C21H25N3O2
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