| 货号:22958-10 mg | 规格:10 mg | 目录价:¥2707 |
| 货号:22958-25 mg | 规格:25 mg | 目录价:¥6244 |
| 货号:22958-5 mg | 规格:5 mg | 目录价:¥1796 |
产品详情
* 以下信息仅供参考,详情请以原厂网站为准
产品名称:
Istradefylline
别名:
KW 6002
产品描述:
An A2A receptor antagonist (Ki = 2.2 nM in a radioligand binding assay); inhibits haloperidol-induced catalepsy (ED50 = 0.23 mg/kg in rats); alleviates postural defects in a dose-dependent manner without inducing dyskinesias or hyperactivity in an MPTP-induced marmoset model of Parkinson's disease; decreases bradykinesias induced by L-DOPA and improves attentional and working memory deficits in an MPTP-induced macaque model of Parkinson's disease
保存温度:
-20
运输温度:
-20
预期分子量:
384.4
产品形式:
A crystalline solid
纯度:
≥98%
CAS号:
155270-99-8
分子式:
C20H24N4O4
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