| 货号:39772-10 mg | 规格:10 mg | 目录价:¥2394 |
| 货号:39772-25 mg | 规格:25 mg | 目录价:¥5320 |
| 货号:39772-5 mg | 规格:5 mg | 目录价:¥1330 |
| 货号:39772-50 mg | 规格:50 mg | 目录价:¥9310 |
产品详情
* 以下信息仅供参考,详情请以原厂网站为准
产品名称:
KB-0742 (hydrochloride)
产品描述:
A Cdk9 inhibitor (IC50 = 6 nM); selective for Cdk9 over Cdk1-8 (IC50s = 397->10,000 nM) and Cdk12-19 (IC50s = 372->10,000 nM); induces cell cycle arrest at the G1 phase and apoptosis in BT-20, BT-549, MDA-MB-231, MT-3, and Hs 578T TNBC cells from 0.64-7.73 µM; reduces tumor volume in the MYC-amplified CTG-0437 PDX mouse model of TNBC at 60 mg/kg
保存温度:
-20
运输温度:
-20
预期分子量:
287.4034
产品形式:
A solid
有效期:
1460
纯度:
≥95%
分子式:
C16H25N5 • HCl
促销活动
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