| 货号:40940-1 mg | 规格:1 mg | 目录价:¥522.6 |
| 货号:40940-10 mg | 规格:10 mg | 目录价:¥4649.8 |
| 货号:40940-25 mg | 规格:25 mg | 目录价:¥10318 |
| 货号:40940-5 mg | 规格:5 mg | 目录价:¥2452.2 |
产品详情
* 以下信息仅供参考,详情请以原厂网站为准
产品名称:
Lirafugratinib
别名:
RLY-4008
产品描述:
A covalent FGFR2 inhibitor (IC50 = 0.003 µM); selective for FGFR2 over FGFR1, -3, and -4 (IC50s = 0.77, 0.26, and 15 µM, respectively); inhibits the proliferation of SNU-16 cells (IC50 = 0.002 µM); reduces intratumoral FGFR2 phosphorylation and tumor volume in an FGFR2-amplified SNU-16 gastric cancer mouse xenograft model at 10 mg/kg
保存温度:
-20
运输温度:
-20
预期分子量:
509.534543
产品形式:
A solid
纯度:
≥98%
CAS号:
2549174-42-5
分子式:
C28H24FN7O2
促销活动
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