| 货号:27056-1 mg | 规格:1 mg | 目录价:¥657 |
| 货号:27056-10 mg | 规格:10 mg | 目录价:¥4100 |
| 货号:27056-25 mg | 规格:25 mg | 目录价:¥9407 |
| 货号:27056-5 mg | 规格:5 mg | 目录价:¥2238 |
产品详情
* 以下信息仅供参考,详情请以原厂网站为准
产品名称:
LOXO-101
别名:
ARRY-470|Larotrectinib
产品描述:
A pan-Trk inhibitor (IC50s = 2-20 nM for TrkA, TrkB, and TrkC); selective for TrkA, -B, and -C over a panel of 226 kinases at 1 μM; inhibits the growth of CUTO-3.29, KM12, and MO-91 patient-derived cancer cell lines (IC50s = <100, <10, and <10 nM, respectively); reduces tumor growth in a KM12 mouse xenograft model at 60 and 200 mg/kg
保存温度:
-20
运输温度:
-20
预期分子量:
428.435426
产品形式:
A crystalline solid
纯度:
≥98%
CAS号:
1223403-58-4
分子式:
C21H22F2N6O2
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