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折扣/货期| 货号：23304-100 mg | 规格：100 mg | 目录价：￥2037 |
| 货号：23304-25 mg | 规格：25 mg | 目录价：￥576 |
| 货号：23304-250 mg | 规格：250 mg | 目录价：￥4462 |
| 货号：23304-50 mg | 规格：50 mg | 目录价：￥1085 |
产品详情
* 以下信息仅供参考，详情请以原厂网站为准
产品名称:
Macitentan
别名:
ACT-064992|Actelion-1
产品描述:
A dual ETA/ETB receptor antagonist (IC50s = 0.5 and 391 nM in a radioligand binding assay using recombinant ETA and ETB, respectively); inhibits ET-1-induced intracellular Ca2+ increase in HPASMCs (IC50 = 0.9 nM) and contractions of isolated rat aortic rings (pA2 = 7.6 for ETA) and sarafotoxin S6c-induced contractions of isolated rat tracheal rings (pA2 = 5.9 for ETB); decreases mean arterial blood pressure in DOCA-salt hypertensive rats (ED50 = 1 mg/kg); prevents development of pulmonary hypertension and right ventricle hypertrophy in a rat model of hypertension; decreases the number of vascular and tubule-interstitial lesions and amount of glomerular damage in a rat model of diabetes
保存温度:
-20
运输温度:
-20
预期分子量:
588.3
产品形式:
A crystalline solid
纯度:
≥98%
CAS号:
441798-33-0
分子式:
C19H20Br2N6O4S
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