| 货号:34477-10 mg | 规格:10 mg | 目录价:¥2774 |
| 货号:34477-25 mg | 规格:25 mg | 目录价:¥5842 |
| 货号:34477-5 mg | 规格:5 mg | 目录价:¥1461 |
产品详情
* 以下信息仅供参考,详情请以原厂网站为准
产品名称:
Nav1.7 Blocker 52
别名:
TC-N 1752|Voltage-gated Sodium Channel 1.7
产品描述:
An inhibitor of Nav1.7 (IC50 = 0.17 µM); selective for Nav1.7 over hERG/Kv11.1, Nav1.5, and Nav1.8 (IC50s = >10, 1.1, and 2.2 µM, respectively) but does inhibit Nav1.3 and Nav1.4 (IC50s = 0.3 and 0.4 µM, respectively); inhibits formalin-induced flinching in a rat model of persistent pain at 20 and 30 mg/kg; increases latency to paw withdrawal in a hot plate test in a mouse model of CFA-induced inflammatory pain
保存温度:
-20
运输温度:
-20
预期分子量:
516.515729
产品形式:
A solid
纯度:
≥98%
CAS号:
1211866-85-1
分子式:
C25H27F3N6O3
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