深圳欣博盛生物科技有限公司 a1

Ocaperidone
货号:42946-10 mg 规格:10 mg 目录价:¥1313
货号:42946-100 mg 规格:100 mg 目录价:¥5923
货号:42946-25 mg 规格:25 mg 目录价:¥1983
货号:42946-50 mg 规格:50 mg 目录价:¥3296
产品详情
* 以下信息仅供参考,详情请以原厂网站为准
产品名称:
Ocaperidone
别名:
R 79598
产品描述:
An atypical antipsychotic; binds to dopamine D2, α1-adrenergic, and 5-HT2 receptors (Kis = 0.75, 0.46, and 0.14 nM, respectively); selective for these receptors over a panel of 26 additional receptors, transporters, channels, and enzymes but does bind to α2-ARs, 5-HT1A, 5-HT1D, and the histamine H1 receptor (Kis = 5.4, 6.8, 9.6, and 1.6 nM, respectively); inhibits apomorphine-induced stereotypy and cocaine- or amphetamine-induced agitation (ED50s = 0.018, 0.042, and 0.014 mg/kg, respectively) and tryptamine-induced clonic seizures and mescaline-induced head twitches (ED50s = 0.021 and 0.037 mg/kg, respectively) in rats; decreases locomotor activity and food intake (ED50s = 0.024 and 0.074 mg/kg, respectively) and induces catalepsy, palpebral ptosis, and hypotonia (ED50s = 0.39, 1.34, and 5.37 mg/kg, respectively) in rats; inhibits LSD-induced drug discrimination, ovalbumin and histamine-induced skin sensitization, acetic acid-induced writhing, and xylazine-induced loss of the righting reflex in rats (ED50s = 0.021, 1.18, 1.34, and 5.37 mg/kg, respectively)
保存温度:
-20
运输温度:
-20
预期分子量:
420.488403
产品形式:
A solid
纯度:
≥95%
CAS号:
129029-23-8
分子式:
C24H25FN4O2
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