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折扣/货期| 货号：43077-1 mg | 规格：1 mg | 目录价：￥965 |
| 货号：43077-10 mg | 规格：10 mg | 目录价：￥6244 |
| 货号：43077-5 mg | 规格：5 mg | 目录价：￥4328 |
产品详情
* 以下信息仅供参考，详情请以原厂网站为准
产品名称:
Orvepitant (maleate)
别名:
GW 823296B
产品描述:
An NK1 receptor antagonist (Ki = 0.06 nM for the human receptor); selective for the NK1 receptor over a panel of 67 transporters, ion channels, and enzymes at 10 µM; inhibits substance P-induced calcium release in CHO cells expressing recombinant human NK1 (apparent pKB = 10.3); inhibits GR73632-induced foot tapping in gerbils (ID50 = 0.11, 0.09, 0.09, and 3.36 mg/kg when administered 1, 4, 8, or 24 hours prior to GR73632, respectively); inhibits GR73632-induced hindlimb scratching in gerbils; reduces the number of territorial postures in the human threat test, indicating anxiolytic-like activity, in marmosets at 1, 3, and 10 mg/kg
保存温度:
-20
运输温度:
-20
预期分子量:
628.635822
产品形式:
A solid
纯度:
≥98%
CAS号:
579475-24-4
分子式:
C31H35F7N4O2 • C4H4O4
促销活动
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