| 货号:21849-1 mg | 规格:1 mg | 目录价:¥724 |
| 货号:21849-5 mg | 规格:5 mg | 目录价:¥2640 |
产品详情
* 以下信息仅供参考,详情请以原厂网站为准
产品名称:
P1075
产品描述:
A potent activator of SUR2-Kir6 and KATP channels; activates SUR2-Kir6 channels (EC50 = 45 nM for SUR2B-Kir6 channel activation); highly selective for SUR2 over SUR1 isoforms (IC50s = 9-46 nM and 1.02 mM, respectively, in a radioligand binding assay); increases outflow facility, a marker of reduced intraocular pressure, in human eye anterior segments ex vivo; reduces infarct size in isolated rabbit hearts via activation of mitochondrial KATP channels (EC50s = 60-90 nM)
保存温度:
-20
运输温度:
-20
预期分子量:
231.3
产品形式:
A crystalline solid
纯度:
≥98%
CAS号:
60559-98-0
分子式:
C12H17N5
促销活动
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