| 货号:16752-10 mg | 规格:10 mg | 目录价:¥1943 |
| 货号:16752-5 mg | 规格:5 mg | 目录价:¥1085 |
| 货号:16752-50 mg | 规格:50 mg | 目录价:¥5293 |
产品详情
* 以下信息仅供参考,详情请以原厂网站为准
产品名称:
Palonosetron (hydrochloride)
别名:
RS 25259-197
产品描述:
A 5-HT3 receptor antagonist (Ki = 0.04 nM); selective for 5-HT3 over 5-HT1A, 5-HT1D, 5-HT2A, and 5-HT2C receptors (Kis = ≥15.85 μM for all), as well as a panel of additional neurotransmitter receptors; inhibits 5-HT-induced contraction in isolated guinea pig ileum; inhibits cisplatin-induced emesis in ferrets (ID50 = 1.1 μg/kg, i.v.); inhibits emesis induced by cisplatin, dacarbazine, actinomycin D, and mechlorethamine in dogs (ID50s = 1.9, 4.1, 4.9, and 4.4 μg/kg, respectively)
保存温度:
-20
运输温度:
-20
预期分子量:
296.44
产品形式:
A crystalline solid
纯度:
≥98%
CAS号:
135729-62-3
分子式:
C19H24N2O • HCl
促销活动
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