| 货号:40142-1 mg | 规格:1 mg | 目录价:¥490 |
| 货号:40142-10 mg | 规格:10 mg | 目录价:¥1960 |
| 货号:40142-25 mg | 规格:25 mg | 目录价:¥3682 |
| 货号:40142-5 mg | 规格:5 mg | 目录价:¥1232 |
产品详情
* 以下信息仅供参考,详情请以原厂网站为准
产品名称:
PF-05190457
产品描述:
An inverse agonist of GHS-R; selectively binds to GHS-R (Ki = 4.37 nM) over M2 mAChRs (Ki = 1,950 nM) and 5-HT2B receptors (IC50 = 3,700 nM); increases glucose-induced insulin secretion in primary human pancreatic islets at 1 µM; potentiates GLP-1-induced intracellular calcium levels in isolated dispersed rat islets at 100 nM; increases ex vivo vagal nerve firing rate in rats when administered intragastrically (EC50 = 10.7 nM)
保存温度:
-20
运输温度:
-20
预期分子量:
512.67022
产品形式:
A solid
有效期:
1460
纯度:
≥95%
CAS号:
1334782-79-4
分子式:
C29H32N6OS
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