深圳欣博盛生物科技有限公司 a1

PF-9363
货号:37778-1 mg 规格:1 mg 目录价:¥590
货号:37778-10 mg 规格:10 mg 目录价:¥4703
货号:37778-25 mg 规格:25 mg 目录价:¥10278
货号:37778-5 mg 规格:5 mg 目录价:¥2653
产品详情
* 以下信息仅供参考,详情请以原厂网站为准
产品名称:
PF-9363
别名:
CTx-648
产品描述:
A KAT6A and KAT6B inhibitor (Kis = 0.27 and 2.4 nM, respectively); selective for KAT6A and KAT6B over KAT7, KAT5, and KAT8 (Kis = 70, 420, and 670 nM, respectively); reduces the proliferation of, and the levels of H3K23Ac and H3K14Ac in, ZR-75-1 cancer cells (IC50s = 0.37, 0.85, and 120 nM, respectively); reduces tumor levels of H3K23Ac and tumor volume without affecting body weight in a ZR-75-1 breast cancer mouse xenograft model at 0.03, 03, or 5 mg/kg per day; reduces tumor volume and increases survival in a PDX mouse model of breast cancer at 1 mg/kg per day
保存温度:
-20
运输温度:
-20
预期分子量:
444.46216
产品形式:
A solid
纯度:
≥98%
CAS号:
2569009-58-9
分子式:
C20H20N4O6S
在线留言
咨询类型
联系人
*
联系方式
*
单位名称
*
咨询内容
*
复制QQ号成功,请打开QQ后添加好友进行咨询