官网链接
折扣/货期| 货号：24192-10 mg | 规格：10 mg | 目录价：￥844 |
| 货号：24192-100 mg | 规格：100 mg | 目录价：￥4864 |
| 货号：24192-250 mg | 规格：250 mg | 目录价：￥10090 |
| 货号：24192-50 mg | 规格：50 mg | 目录价：￥2854 |
产品详情
* 以下信息仅供参考，详情请以原厂网站为准
产品名称:
Prucalopride
产品描述:
A potent and selective 5-HT4 agonist (Ki = 2.5 and 8 nM for 5-HT4A and 5-HT4B, respectively); greater than 250-fold selective for 5-HT4 over a panel of 53 overexpressed receptors, including 5-HT subtypes, but does bind to human D4 and σ1 receptors and mouse 5-HT3 receptors (Kis = 2.3, 3.7, and 3.8 μM respectively); induces 5-HT4-dependent contractions in guinea pig colon (EC50 = 33 nM) and facilitates non-cholinergic contractions induced by electrical stimulation; increases colonic motility by inhibiting distal colon contractions in dogs (ED50 = 0.04 mg/kg, p.o.); increases acetylcholine and histamine levels in the rat prefrontal cortex and the power of hippocampal theta oscillations (5-10 mg/kg, s.c.)
保存温度:
-20
运输温度:
-20
产品形式:
A crystalline solid
纯度:
≥98%
CAS号:
179474-81-8
分子式:
C18H26ClN3O3
促销活动
精品推荐
复制QQ号成功，请打开QQ后添加好友进行咨询