| 货号:21203-1 mg | 规格:1 mg | 目录价:¥844 |
| 货号:21203-10 mg | 规格:10 mg | 目录价:¥5668 |
| 货号:21203-5 mg | 规格:5 mg | 目录价:¥3243 |
产品详情
* 以下信息仅供参考,详情请以原厂网站为准
产品名称:
PX-13-17OH
产品描述:
A PI3K inhibitor; inhibits PI3Kα, PI3Kβ, PI3Kɣ, and PI3Kδ (IC50s = 6.4, 13, 8, and 11 nM, respectively) over mTOR (IC50 = 2.9 µM); 420-fold selective for PI3K in a panel of 20 lipid and protein kinases; inhibits phosphorylation of Akt and S6K in PTEN-negative U87MG cells at 0.03-1 µg/ml; inhibits tumor growth in a U87MG mouse xenograft model at 2.5-10 mg/kg
保存温度:
-20
运输温度:
-20
预期分子量:
546.7
产品形式:
A crystalline solid
纯度:
≥98%
CAS号:
884539-95-1
分子式:
C29H42N2O8
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