| 货号:26231-1 mg | 规格:1 mg | 目录价:¥1849.2 |
| 货号:26231-10 mg | 规格:10 mg | 目录价:¥11055 |
| 货号:26231-5 mg | 规格:5 mg | 目录价:¥8308 |
产品详情
* 以下信息仅供参考,详情请以原厂网站为准
产品名称:
QC6352
产品描述:
A KDM4 inhibitor; selective for KDM4A, KDM4B, KDM4C, and KDM4D (IC50s = 104, 56, 35, and 104 nM, respectively) over KDM2B, KDM3A, KDM3B, KDM6B, and PHF8 (IC50s = >4,000 nM for all) but does inhibit KDM5B (IC50 = 750 nM); increases H3K36Me3 levels in KYSE-150 cells (EC50 = 1.3 nM); reduces the proliferation of KYSE-150 cells (EC50 = 3.5 nM) but not IMR-90 fibroblasts (IC50 = >30 µM); reduces tumor volume in a BR0859f PDX mouse model of HER2-positive breast cancer at 10, 25, and 50 mg/kg
保存温度:
-20
运输温度:
-20
预期分子量:
387.47432
产品形式:
A solid
有效期:
1460
纯度:
≥98%
CAS号:
1851373-36-8
分子式:
C24H25N3O2
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