| 货号:21221-1 mg | 规格:1 mg | 目录价:¥482 |
| 货号:21221-10 mg | 规格:10 mg | 目录价:¥3162 |
| 货号:21221-25 mg | 规格:25 mg | 目录价:¥5628 |
| 货号:21221-5 mg | 规格:5 mg | 目录价:¥1715 |
产品详情
* 以下信息仅供参考,详情请以原厂网站为准
产品名称:
R-59-949
别名:
Diacylglycerol Kinase Inhibitor II|DKGI-II
产品描述:
A DGK-α inhibitor (IC50 = 300 nM in isolated platelet plasma membranes); increases diacylglycerol-dependent PKC activity, serotonin secretion, and aggregation of thrombin-stimulated platelets; inhibits PDGF-induced DGK-α activity in intact VSMCs; inhibits high K+- and glucose-induced insulin secretion in MIN6 pancreatic β-cells in a dose-dependent manner; prevents retinal neovascularization in a mouse model of oxygen-induced retinopathy
保存温度:
-20
运输温度:
-20
预期分子量:
489.6
产品形式:
A crystalline solid
纯度:
≥98%
CAS号:
120166-69-0
分子式:
C28H25F2N3OS
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