| 货号:36890-1 mg | 规格:1 mg | 目录价:¥3082 |
| 货号:36890-10 mg | 规格:10 mg | 目录价:¥16951 |
| 货号:36890-5 mg | 规格:5 mg | 目录价:¥10800.4 |
产品详情
* 以下信息仅供参考,详情请以原厂网站为准
产品名称:
R 715 (trifluoroacetate salt)
别名:
[Ac-Lys-[D-βNal7,Ile8]des-Arg9]-BK|Ac-Lys-Arg-Pro-Pro-Gly-Phe-Ser-D2Nal-Ile-OH
产品描述:
A bradykinin B1 receptor antagonist; inhibits bradykinin-induced contractions in isolated human umbilical cords, which express bradykinin B1 receptors (pA2 = 8.49); decreases the latency to tail withdrawal in the tail-flick test in an STZ-induced mouse model of diabetic neuropathy at 200, 400, and 600 µg/kg; reduces the incidence of hind limb weakness and paralysis, improves symmetrical gait, as well as decreases spinal inflammatory foci numbers, neuron demyelination, and lesion monocyte invasion, in a MOG35-55 peptide-induced mouse model of EAE at 1 mg/kg per day; reduces mean arterial blood pressure and increases heart rate in spontaneously hypertensive rats at 0.01 nmol/animal, i.c.v
保存温度:
-20
运输温度:
-20
预期分子量:
1140.33346
产品形式:
A solid
有效期:
1460
纯度:
≥95%
分子式:
C57H81N13O12 • XCF3COOH
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