| 货号:23697-10 mg | 规格:10 mg | 目录价:¥1126 |
| 货号:23697-25 mg | 规格:25 mg | 目录价:¥2184 |
| 货号:23697-5 mg | 规格:5 mg | 目录价:¥590 |
| 货号:23697-50 mg | 规格:50 mg | 目录价:¥4074 |
产品详情
* 以下信息仅供参考,详情请以原厂网站为准
产品名称:
Saxagliptin (hydrochloride)
别名:
BMS-477118
产品描述:
A potent DPP-4 inhibitor (Ki = 0.6 nM); inhibits DPP-4 ex vivo (ED50 = 0.12 μmol/kg) in plasma from normal fasted rats; reduces plasma glucose levels in Zuckerfa/fa diabetic rats in a dose-dependent manner when administered orally in doses ranging from 0.3-3 mg/kg; increases plasma insulin levels and improves glucose clearance in ob/ob mice; induces systolic and diastolic dysfunction, reduces contractile force, and exacerbates ischemia-reperfusion injury-induced cardiac dysfunction in isolated guinea pig hearts
保存温度:
-20
运输温度:
-20
预期分子量:
315.44
产品形式:
A crystalline solid
纯度:
≥98%
CAS号:
709031-78-7
分子式:
C18H25N3O2 • HCl
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