| 货号:36217-1 mg | 规格:1 mg | 目录价:¥657 |
| 货号:36217-5 mg | 规格:5 mg | 目录价:¥1956 |
产品详情
* 以下信息仅供参考,详情请以原厂网站为准
产品名称:
SB-243213 (hydrochloride)
产品描述:
A 5-HT2C receptor inverse agonist; selective for 5-HT2C over the 5-HT2A and 5-HT2B receptors (Kis = 0.001, 0.158, and 0.1 µM, respectively) and CYP1A2, CYP2C9, CYP2C19, CYP2D6, and CYP3A4 (IC50s = >100, 23, >100, >100, and >100 µM, respectively); reduces the basal activity of 5-HT2C in HEK293 cells expressing the human receptor (pKB = 9.5); reverses mCPP-induced hypolocomotion in rats (ID50 = 0.7 mg/kg); has anxiolytic-like activity in the social interaction test in rats at 0.2-5 mg/kg
保存温度:
-20
运输温度:
-20
预期分子量:
428.407229
产品形式:
A solid
纯度:
≥98%
CAS号:
1780372-25-9
分子式:
C22H19F3N4O2 • 2HCl
促销活动
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