| 货号:27338-10 mg | 规格:10 mg | 目录价:¥1581 |
| 货号:27338-25 mg | 规格:25 mg | 目录价:¥3444 |
| 货号:27338-5 mg | 规格:5 mg | 目录价:¥844 |
| 货号:27338-50 mg | 规格:50 mg | 目录价:¥6445 |
产品详情
* 以下信息仅供参考,详情请以原厂网站为准
产品名称:
Sitravatinib
别名:
MGCD-516
产品描述:
A multi-kinase inhibitor; inhibits 35 kinases (IC50s = 0.5-4,098 nM) in a panel of 55 RTKs; reduces proliferation in various cancer cells (IC50s = 340.1-1,830 nM) and decreases phosphorylation of IGF1-R, PDGFRβ, and Akt at 62.5-4,000 nM; decreases tumor growth in LPS141 and MPNST mouse xenograft models at 15 mg/kg per day
保存温度:
-20
运输温度:
-20
预期分子量:
629.677466
产品形式:
A crystalline solid
纯度:
≥98%
CAS号:
1123837-84-2
分子式:
C33H29F2N5O4S
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