| 货号:14974-1 mg | 规格:1 mg | 目录价:¥1206 |
| 货号:14974-10 mg | 规格:10 mg | 目录价:¥3564.4 |
| 货号:14974-5 mg | 规格:5 mg | 目录价:¥2117.2 |
| 货号:14974-50 mg | 规格:50 mg | 目录价:¥11550.8 |
产品详情
* 以下信息仅供参考,详情请以原厂网站为准
产品名称:
SNS-314 (mesylate)
产品描述:
A pan-Aurora kinase inhibitor (IC50s = 9, 31, and 3.4 nM for Aurora A, B, and C, respectively); inhibits TRKB, TRKA, FLT4, FMS, DDR2, AXL, and C-RAF (IC50s = 5-100 nM); inhibits Aurora B phosphorylation of histone H3 in HCT116 human colorectal carcinoma cells in vitro (EC50 = <16 nM) and in a mouse xenograft model at a dose of 50 mg/kg; inhibits tumor growth in A2780 ovarian, A375 melanoma, H1299 lung, MDA-MB-231 breast, and PC3 prostate cancer mouse xenograft models
保存温度:
-20
运输温度:
-20
预期分子量:
527
产品形式:
A crystalline solid
有效期:
1460
纯度:
≥98%
CAS号:
1146618-41-8
分子式:
C18H15ClN6OS2 • CH3SO3H
促销活动
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