| 货号:39811-1 mg | 规格:1 mg | 目录价:¥576.2 |
| 货号:39811-10 mg | 规格:10 mg | 目录价:¥4328.2 |
| 货号:39811-5 mg | 规格:5 mg | 目录价:¥2599.6 |
产品详情
* 以下信息仅供参考,详情请以原厂网站为准
产品名称:
ST1936
产品描述:
A 5-HT6 receptor agonist; selectively binds to 5-HT6 (Ki = 31 nM) over 5-HT1A, 5-HT1B, 5-HT1D, 5-HT2A, 5-HT2B, 5-HT2C, 5-HT3, 5-HT4, 5-HT5A, and SERT (Kis = >1,000 nM for all) but also binds to the 5-HT7 receptor (Ki = 168 nM); induces cAMP accumulation in BHK fibroblasts (EC50 = 16 nM); decreases the basal firing rate of dopaminergic neurons in the ventral tegmental area but not substantia nigra pars compacta in rats; prevents stress-induced decreases in vanilla sugar-sustained appetitive behavior, indicating anti-anhedonic-like activity, in rats at 10 and 30 mg/kg; induces self-administration in rats at 1 mg/kg
保存温度:
-20
运输温度:
-20
预期分子量:
236.74026
产品形式:
A solid
有效期:
1460
纯度:
≥98%
CAS号:
1210-81-7
分子式:
C13H17ClN2
促销活动
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