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折扣/货期| 货号：11984-1 mg | 规格：1 mg | 目录价：￥482.4 |
| 货号：11984-10 mg | 规格：10 mg | 目录价：￥2720.2 |
| 货号：11984-5 mg | 规格：5 mg | 目录价：￥1474 |
产品详情
* 以下信息仅供参考，详情请以原厂网站为准
产品名称:
Sumanirole (maleate)
别名:
PNU 95666
产品描述:
A dopamine D2 receptor agonist; selective for D2 over D1, D3, and D4 receptors (Kis = 9.0, >7,140, 1,940, and >2,190 nM, respectively); inhibits forskolin-stimulated cAMP accumulation in CHO cells expressing human recombinant D2A receptors (EC50 = 17 nM); decreases plasma prolactin levels in rats at ≥3.1 µmol/kg; inhibits dopamine neuron firing in the SNPC in anesthetized rats (ED50 = 2.3 µmol/kg); increases horizontal locomotor activity in a reserpinized, AMPT rat model of Parkinson's disease at ≥12.5 µmol/kg; decreases time spent in the open arms of the elevated plus maze and time spent immobile in the forced swim test in mice with SNPC lesions at 0.1 mg/kg; reduces premature responding by rats in the 5CRTT compared with untreated animals at ≥0.1 mg/kg
保存温度:
-20
运输温度:
-20
预期分子量:
319.3
产品形式:
A crystalline solid
有效期:
1460
纯度:
≥98%
CAS号:
179386-44-8
分子式:
C11H13N3O • C4H4O4
促销活动
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