Tadalafil-抑制剂-深圳欣博盛生物科技有限公司

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Tadalafil

品牌：Adipogen

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说明书

折扣/货期

货号：CDX-T0455-M050	规格：50 mg	目录价：￥1022
货号：CDX-T0455-M500	规格：500 mg	目录价：￥6440

产品详情

* 以下信息仅供参考，详情请以原厂网站为准

产品名称:

Tadalafil

别名:

GF196960; (6R,12aR)-6-(1,3-Benzodioxol-5-yl)-2,3,6,7,12,12a-hexahydro-2-methylpyrazino[1,2:1,6]pyrido[3,4-b]indole-1,4-dione

产品描述:

Tadalafil is a potent long-acting and selective inhibitor of the cGMP specific phosphodiesterase 5 (PDE5; IC50 = 1.2 nM). It is selective for PDE5 over PDE1-4 and 7-10 (IC50s = 9.2-280 µM), however, it does also inhibit PDE11 (IC50 = 11 nM). In vivo, tadalafil (10 mg/kg) decreases production of the proinflammatory cytokines TNF-alpha, IL-1beta, and IL-6 and improves renal function in a rat model of ischemia/reperfusion injury. Formulations containing tadalafil have been used to treat erectile dysfunction, pulmonary arterial hypertension, benign prostatic hyperplasia (BPH) and lower urinary tract dysfunction. Also delays tumor growth in a mouse model via inhibition of MDSC-mediated immunosuppression.

保存温度:

-20°C

运输温度:

Ambient

预期分子量:

389.4

产品形式:

solid

产地:

瑞士

纯度:

>98%