深圳欣博盛生物科技有限公司 a1

Talarozole
货号:42372-10 mg 规格:10 mg 目录价:¥2399
货号:42372-25 mg 规格:25 mg 目录价:¥4208
货号:42372-5 mg 规格:5 mg 目录价:¥1407
货号:42372-50 mg 规格:50 mg 目录价:¥5601
产品详情
* 以下信息仅供参考,详情请以原厂网站为准
产品名称:
Talarozole
别名:
R115866|Rambazole
产品描述:
A CYP26 inhibitor (IC50 = 0.004 µM); selective for CYP26 over CYP2A1, CYP2C11, CYP17, and CYP19 (IC50s = 9.1, 7.2, 2.6, and 1.3 µM, respectively); increases the levels of all-trans retinoic acid in plasma, skin, liver, fat, kidneys, and spleen in rats at 2.5 mg/kg; inhibits estrogen-induced vaginal keratinization in ovariectomized rats (ED50 = 1 mg/kg), an effect that can be reversed by AGN 193109; increases pinnal epidermal thickness and tail epidermal orthokeratosis percentage in mice from 0.6-2.6 mg/kg
保存温度:
-20
运输温度:
-20
预期分子量:
377.50702
产品形式:
A solid
纯度:
≥95%
CAS号:
201410-53-9
分子式:
C21H23N5S
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