深圳欣博盛生物科技有限公司 a1

TC 2559 (fumarate)
货号:25600-1 mg 规格:1 mg 目录价:¥482
货号:25600-10 mg 规格:10 mg 目录价:¥3390
货号:25600-25 mg 规格:25 mg 目录价:¥7866
货号:25600-5 mg 规格:5 mg 目录价:¥2050
产品详情
* 以下信息仅供参考,详情请以原厂网站为准
产品名称:
TC 2559 (fumarate)
产品描述:
A partial agonist for α4β2 subunit-containing nAChRs (EC50 = 0.18 µM); selective for α4β2 over α2β4, α4β4, α3β4, α3β2, and α7 subunit-containing nAChRs (EC50s = 14, 12.5, >30, >100, and >100 µM, respectively); increases dopamine cell firing in the rat VTA in vitro; enhances inhibitory synaptic transmission in dorsal horn neurons via α4β2 subunit-containing nAChRs; reduces formalin-induced paw-licking time in mice at 3 and 10 mg/kg; reverses scopolamine-induced cognitive deficits in rats in a step-through passive avoidance test at 3 and 6 µmol/kg
保存温度:
-20
运输温度:
-20
预期分子量:
206.2842
产品形式:
A solid
纯度:
≥95%
CAS号:
212332-35-9
分子式:
C12H18N2O • 2C4H4O4
在线留言
咨询类型
联系人
*
联系方式
*
单位名称
*
咨询内容
*
复制QQ号成功,请打开QQ后添加好友进行咨询