深圳欣博盛生物科技有限公司 a1

TD-4208
货号:36549-10 mg 规格:10 mg 目录价:¥536
货号:36549-100 mg 规格:100 mg 目录价:¥2908
货号:36549-25 mg 规格:25 mg 目录价:¥1072
货号:36549-50 mg 规格:50 mg 目录价:¥1729
产品详情
* 以下信息仅供参考,详情请以原厂网站为准
产品名称:
TD-4208
别名:
Revefenacin
产品描述:
An antagonist of muscarinic acetylcholine receptors (Kis = 0.42, 0.3, 0.18, and 0.55 nM for M1, M2, M3, and M4 receptors, respectively, in CHO-K1 cell membranes with the human receptors); selective for these receptors over M5 muscarinic receptors (Ki = 6.31 nM in CHO-K1 cell membranes with the human receptor); inhibits AChE-induced calcium mobilization in CHO-K1 cells expressing M2 and M3 muscarinic receptors; decreases AChE-induced contractions in isolated rat trachea in a concentration-dependent manner; decreases AChE-induced bronchoconstriction and reduces pilocarpine-induced salivation, a surrogate test for noisy breathing, in rats (ID50s = 45 and 1,164 µg/ml, respectively); decreases AChE-induced bronchoconstriction in dogs at 10 and 30 µg/kg intranasally
保存温度:
-20
运输温度:
-20
预期分子量:
597.8
产品形式:
A solid
纯度:
≥98%
CAS号:
864750-70-9
分子式:
C35H43N5O4
在线留言
咨询类型
联系人
*
联系方式
*
单位名称
*
咨询内容
*
复制QQ号成功,请打开QQ后添加好友进行咨询