深圳欣博盛生物科技有限公司 a1

TG 100-115
货号:10010512-1 mg 规格:1 mg 目录价:¥375
货号:10010512-10 mg 规格:10 mg 目录价:¥2586
货号:10010512-5 mg 规格:5 mg 目录价:¥1568
货号:10010512-50 mg 规格:50 mg 目录价:¥5990
产品详情
* 以下信息仅供参考,详情请以原厂网站为准
产品名称:
TG 100-115
产品描述:
A PI3Kγ and PI3Kδ inhibitor (IC50s = 0.083 and 0.235 µM, respectively); selective for PI3Kγ and PI3Kδ over PI3Kα and PI3Kβ (IC50s = 1.3 and 1.2 µM); inhibits TRPM7 kinase activity (IC50 = 1.07 µM); inhibits the migration and invasion of MDA-MB-231 breast cancer cells at 50 µM; prevents VEGF- or histamine-induced intradermal edema and PAF- or dextran-induced hind paw edema and leukocyte infiltration in rats at 1 and 5 mg/kg, respectively; decreases infarct size as a percentage of the area at risk in a porcine model of myocardial infarction induced by coronary artery occlusion at 0.5 mg/kg
保存温度:
-20
运输温度:
-20
预期分子量:
346.3
产品形式:
A crystalline solid
纯度:
≥95%
CAS号:
677297-51-7
分子式:
C18H14N6O2
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