| 货号:26386-1 mg | 规格:1 mg | 目录价:¥657 |
| 货号:26386-10 mg | 规格:10 mg | 目录价:¥7035 |
| 货号:26386-25 mg | 规格:25 mg | 目录价:¥10211 |
| 货号:26386-5 mg | 规格:5 mg | 目录价:¥3980 |
产品详情
* 以下信息仅供参考,详情请以原厂网站为准
产品名称:
THZ531
产品描述:
An inhibitor of Cdk12 and Cdk13 (IC50s = 158 and 69 nM for Cdk12/cyclin K and Cdk13/cyclin K, respectively); selective for Cdk12/cyclin K and Cdk13/cyclin K over Cdk9/cyclin T1 and Cdk7/cyclin H/MAT1 (IC50s = 10.5 and 8.5 μM, respectively); inhibits proliferation of Jurkat cells (IC50 = 50 nM); induces apoptosis in Jurkat cells in a concentration-dependent manner; reduces expression of genes associated with the DNA damage response, including BRCA1, FANCF, and ERCC4, in Jurkat cells at 50 nM
保存温度:
-20
运输温度:
-20
预期分子量:
558.07376
产品形式:
A crystalline solid
纯度:
≥95%
CAS号:
1702809-17-3
分子式:
C30H32ClN7O2
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