| 货号:26184-1 mg | 规格:1 mg | 目录价:¥482 |
| 货号:26184-10 mg | 规格:10 mg | 目录价:¥3591 |
| 货号:26184-5 mg | 规格:5 mg | 目录价:¥2050 |
产品详情
* 以下信息仅供参考,详情请以原厂网站为准
产品名称:
CC-671
产品描述:
A dual inhibitor of Mps1/TTK and Clk2 (IC50s = 5 and 3 nM, respectively); selective for Mps1/TTK and Clk2 over a panel of 255 kinases at 3 μM; inhibit DYRK3, DYRK1A, PHKG, DYRK1B, and Clk1 (IC50s = 99, 104, 136, 157, and 300 nM, respectively); selectively inhibits the growth of Cal-51 TNBC cell over BT-474 luminal breast cancer cells (IC50s = 60 and 6,970 nM, respectively); reduces tumor volume in a Cal-51 mouse xenograft model at 20 mg/kg
保存温度:
-20
运输温度:
-20
预期分子量:
512.55996
产品形式:
A crystalline solid
纯度:
≥95%
CAS号:
1618658-88-0
分子式:
C28H28N6O4
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