深圳欣博盛生物科技有限公司 a1

Ciproxifan (maleate)
货号:29513-1 mg 规格:1 mg 目录价:¥496
货号:29513-10 mg 规格:10 mg 目录价:¥3296
货号:29513-25 mg 规格:25 mg 目录价:¥6419
货号:29513-5 mg 规格:5 mg 目录价:¥1769
产品详情
* 以下信息仅供参考,详情请以原厂网站为准
产品名称:
Ciproxifan (maleate)
别名:
FUB-359
产品描述:
A histamine H3 receptor antagonist (Ki = 0.5 nM for inhibition of histamine release in rat synaptosomal preparations); selective for histamine H3 over histamine H1 and H2, M3 muscarinic, and α1D- and β1-adrenergic receptors (Kis = 3.15-25 µM), as well as 5-HT1B, 5-HT2A, 5-HT3, and 5-HT4 (Kis = 1.58-15 µM) in radioligand binding assays; inhibits R-(–)-α-methylhistamine-induced relaxation in precontracted isolated guinea pig ileal longitudinal muscle from 3-300 nM; reduces R-(–)-α-methylhistamine-induced water consumption in rats (ED50 = 0.09 mg/kg); increases wake episode duration and latency to fall asleep in rats when administered at a dose of 2 mg/kg
保存温度:
-20
运输温度:
-20
预期分子量:
270.3264
产品形式:
A crystalline solid
纯度:
≥98%
CAS号:
184025-19-2
分子式:
C16H18N2O2 • C4H4O4
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